SCHEMBL2858191

SCHEMBL2858191

COc1cc(CNC(=O)c2cnn(-c3ccc(F)cc3)c2C(F)(F)F)cc(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 8/20 0.56
DGAT2 Q96PD7 2/20 0.51
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TRPC3 Q13507 1/20 0.46
P2RX7 Q99572 1/20 0.46
RORC P51449 1/20 0.46
TP53 P04637 2/20 0.45
DDR1 Q08345 1/20 0.45
MAPK11 Q15759 1/20 0.45
MAPK14 Q16539 1/20 0.45
DDR2 Q16832 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
MAP3K20 Q9NYL2 1/20 0.45
MAP3K2 Q9Y2U5 1/20 0.45
NR3C1 P04150 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856127 0.91 CCR1 (0.64) CCR1DGAT2TP53
SCHEMBL2852791 0.91 CCR1 (0.57) CCR1DGAT2KDM4EALDH1A1TRPC3
SCHEMBL2855224 0.91 CCR1 (0.55) CCR1DGAT2KDM4EALDH1A1RORC
SCHEMBL2855701 0.86 CCR1 (0.54) CCR1DGAT2KDM4EALDH1A1TRPC3
SCHEMBL2857923 0.85 CCR1 (0.66) CCR1KDM4EALDH1A1TRPC3P2RX7
SCHEMBL2850896 0.85 DGAT2 (0.57) CCR1DGAT2KDM4EALDH1A1P2RX7
SCHEMBL2856797 0.84 P2RX7 (0.45) CCR1ALDH1A1P2RX7NR3C1
SCHEMBL2857267 0.84 CCR1 (0.63) CCR1KDM4EALDH1A1TRPC3P2RX7
SCHEMBL2850316 0.84 TP53 (0.59) CCR1DGAT2KDM4EALDH1A1TP53
SCHEMBL2857342 0.83 CCR1 (0.60) CCR1KDM4EALDH1A1TRPC3DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed