SCHEMBL2859504

SCHEMBL2859504

O=C(NCCc1ccc(Cl)cc1)Oc1cnn(-c2cccc(Cl)n2)c1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.43
CNR1 P21554 2/20 0.39
TRPA1 O75762 1/20 0.38
MAPT P10636 3/20 0.37
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.36
HKDC1 Q2TB90 1/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SCN2A Q99250 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854467 0.94 MAPT (0.36) TAAR1CNR1MAPTLMNATRPV1
SCHEMBL2859594 0.88 TAAR1 (0.45) TAAR1CNR1TRPA1MAPTGPBAR1
SCHEMBL2850252 0.88 TRPV1 (0.40) CNR1LMNATRPV1
SCHEMBL2860669 0.86 TAAR1 (0.46) TAAR1CNR1MAPTHRH4HRH3
SCHEMBL2859861 0.85 TAAR1 (0.51) TAAR1CNR1MAPTLMNACYP1A2
SCHEMBL2857979 0.85 TRPV1 (0.39) TAAR1CNR1MEN1KMT2AHSD17B10
SCHEMBL2853336 0.85 TAAR1 (0.45) TAAR1CNR1TRPA1MAPTHRH4
SCHEMBL2853347 0.84 TRPV1 (0.41) MAPTCCR1TRPV1
SCHEMBL2855547 0.83 TAAR1 (0.54) TAAR1CNR1MAPTLMNACCR1
SCHEMBL2860458 0.83 TP53 (0.46) TAAR1CNR1MAPTLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed