SCHEMBL2861643

SCHEMBL2861643

COc1ccc(-n2ncc(OC(=O)NCCc3ccc(Cl)cc3)c2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.50
FPR2 P25090 1/20 0.50
KMT2A Q03164 5/20 0.49
GLA P06280 1/20 0.49
TAAR1 Q96RJ0 2/20 0.48
NPC1 O15118 1/20 0.48
GAA P10253 1/20 0.48
RAB9A P51151 1/20 0.48
MEN1 O00255 1/20 0.47
TP53 P04637 1/20 0.47
ALDH1A1 P00352 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
POLB P06746 1/20 0.44
ATM Q13315 1/20 0.43
ABCB1 P08183 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853389 0.90 NPC1 (0.62) FPR2KMT2AGLATAAR1NPC1
SCHEMBL2854531 0.90 LMNA (0.52) KMT2ANPC1RAB9AMEN1TP53
SCHEMBL2854313 0.89 NPSR1 (0.54) CNR1TAAR1TP53LMNA
SCHEMBL2859872 0.89 TAAR1 (0.54) KMT2ATAAR1NPC1GAARAB9A
SCHEMBL2857343 0.87 P2RX7 (0.42) CNR1KMT2AMEN1TP53ALDH1A1
SCHEMBL2858680 0.84 NPC1 (0.45) KMT2ATAAR1NPC1GAARAB9A
SCHEMBL2856862 0.83 NPC1 (0.53) KMT2ATAAR1NPC1GAARAB9A
SCHEMBL2857468 0.83 MAPT (0.47) NPC1RAB9ATP53ALDH1A1SMN1; SMN2
SCHEMBL2852384 0.82 NPC1 (0.54) CNR1KMT2ANPC1GAARAB9A
SCHEMBL2850323 0.82 MAPT (0.47) KMT2AGLATAAR1NPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed