SCHEMBL2858680

SCHEMBL2858680

COc1ccc(-n2ncc(OC(=O)NCCc3ccccc3Cl)c2C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
MAPT P10636 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
GAA P10253 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
PKM P14618 1/20 0.43
ABCB11 O95342 1/20 0.43
P2RX7 Q99572 1/20 0.43
KMT2A Q03164 2/20 0.43
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
NPBWR1 P48145 4/20 0.41
TP53 P04637 2/20 0.40
MCHR1 Q99705 2/20 0.40
S1PR4 O95977 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856602 0.91 RIPK1 (0.46) MAPTABCB11P2RX7KMT2ATP53
SCHEMBL2850323 0.90 MAPT (0.47) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL2853335 0.90 TP53 (0.48) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL2857343 0.89 P2RX7 (0.42) MAPTSMN1; SMN2P2RX7KMT2ANPBWR1
SCHEMBL2853389 0.86 NPC1 (0.62) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL2861643 0.84 CNR1 (0.50) NPC1RAB9ASMN1; SMN2GAATAAR1
SCHEMBL2860652 0.83 POLB (0.44) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL2851589 0.82 MTNR1A (0.48) MAPTSMN1; SMN2KMT2ATP53ALDH1A1
SCHEMBL2854704 0.82 P2RX7 (0.48) MAPTSMN1; SMN2PKMP2RX7KMT2A
SCHEMBL2856862 0.82 NPC1 (0.53) NPC1RAB9AMAPTSMN1; SMN2NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed