SCHEMBL2862272

SCHEMBL2862272

Cc1c(OC(=O)NCCc2cccc(C(F)(F)F)c2)cnn1-c1ccc(F)cc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 14/20 0.61
NPSR1 Q6W5P4 2/20 0.58
KDM4E B2RXH2 1/20 0.58
MAPT P10636 2/20 0.49
HSP90AA1 P07900 1/20 0.49
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
CNR1 P21554 1/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854340 0.90 CCR1 (0.53) CCR1NPSR1KDM4EMAPTHSP90AA1
SCHEMBL2857365 0.87 CCR1 (0.49) CCR1NPSR1KDM4EMAPT
SCHEMBL2853261 0.86 SPR (0.48) CCR1NPSR1KDM4EMAPT
SCHEMBL2857468 0.85 MAPT (0.47) CCR1NPSR1KDM4EMAPT
SCHEMBL2854225 0.83 CCR1 (0.60) CCR1NPSR1KDM4EMAPTHSP90AA1
SCHEMBL2862820 0.82 P2RX7 (0.45) CCR1NPSR1KDM4EMAPTCNR1
SCHEMBL2863198 0.82 CCR1 (0.50) CCR1NPSR1KDM4EMAPTROCK2
SCHEMBL2857735 0.82 CCR1 (0.54) CCR1NPSR1KDM4EMAPTHSP90AA1
SCHEMBL2854313 0.81 NPSR1 (0.54) CCR1NPSR1MAPTCNR1
SCHEMBL2860847 0.81 CCR1 (0.55) CCR1NPSR1KDM4EMAPTHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed