SCHEMBL2853261

SCHEMBL2853261

COc1cccc(CCNC(=O)Oc2cnn(-c3ccc(F)cc3)c2C)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.48
TDP1 Q9NUW8 1/20 0.46
SMO Q99835 1/20 0.46
CCR1 P32246 1/20 0.44
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852556 0.88 TDP1 (0.44) SPRTDP1CCR1MAPTTP53
SCHEMBL2857365 0.88 CCR1 (0.49) CCR1MAPTTP53NPC1RAB9A
SCHEMBL2862272 0.86 CCR1 (0.61) CCR1MAPTKDM4ENPSR1
SCHEMBL2857468 0.86 MAPT (0.47) SPRSMOCCR1MAPTTP53
SCHEMBL2853389 0.84 NPC1 (0.62) MAPTTP53NPC1RAB9AALDH1A1
SCHEMBL2851589 0.83 MTNR1A (0.48) MAPTTP53ALDH1A1
SCHEMBL2854313 0.82 NPSR1 (0.54) SPRTDP1CCR1MAPTTP53
SCHEMBL2854586 0.81 ALDH1A1 (0.47) SPRMAPTNPC1RAB9AALDH1A1
SCHEMBL2854802 0.81 LMNA (0.48) CCR1MAPTTP53ALDH1A1POLB
SCHEMBL2863131 0.80 CNR1 (0.50) SPRCCR1MAPTTAAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed