SCHEMBL2862974

SCHEMBL2862974

CS(=O)(=O)c1cccc(NC(=O)Oc2cnn(-c3ccccc3)c2C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.50
NFE2L2 Q16236 2/20 0.50
BRAF P15056 1/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CARM1 Q86X55 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
EPHX2 P34913 1/20 0.41
PTGS2 P35354 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 2/20 0.40
CSNK2A1 P68400 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MET P08581 1/20 0.40
MST1R Q04912 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856385 0.93 CCR1 (0.44) KEAP1NFE2L2BRAFCARM1EPHX2
SCHEMBL2855798 0.92 MAPT (0.45) KEAP1NFE2L2MAPTSMN1; SMN2KMT2A
SCHEMBL2855716 0.92 KEAP1 (0.46) KEAP1NFE2L2BRAFPOLBMAPT
SCHEMBL2856588 0.92 KEAP1 (0.42) KEAP1NFE2L2BRAFMAPTSMN1; SMN2
SCHEMBL2853595 0.90 LMNA (0.44) KEAP1NFE2L2MAPTSMN1; SMN2KDM4E
SCHEMBL2869545 0.89 KEAP1 (0.40) KEAP1NFE2L2BRAFMAPTSMN1; SMN2
SCHEMBL2860990 0.89 KEAP1 (0.43) KEAP1NFE2L2MAPTKMT2ACARM1
SCHEMBL2852487 0.89 MAPT (0.48) KEAP1NFE2L2MAPTSMN1; SMN2KMT2A
SCHEMBL2854592 0.88 MEN1 (0.40) KEAP1NFE2L2MAPTSMN1; SMN2KMT2A
SCHEMBL2861567 0.87 MALT1 (0.41) KEAP1NFE2L2MAPTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed