SCHEMBL286414

SCHEMBL286414

CCCCc1noc(C)c1COc1cc(C(=O)OC(CO)C(N)=O)[nH]n1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 11/20 0.32
GABRA5 P31644 4/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.30
ALPL P05186 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286582 0.91 KMT2A (0.38) GABRA1GABRA5L3MBTL1ALDH1A1KMT2A
SCHEMBL286328 0.91 KMT2A (0.38) GABRA1GABRA5L3MBTL1ALDH1A1KMT2A
SCHEMBL286463 0.85 ALDH1A1 (0.34) GABRA1GABRA5L3MBTL1ALDH1A1KMT2A
SCHEMBL286460 0.85 ALPL (0.43) GABRA5L3MBTL1ALDH1A1KMT2AALPL
SCHEMBL286337 0.83 HCAR2 (0.39) GABRA5L3MBTL1ALPL
SCHEMBL286162 0.82 GABRA5 (0.43) GABRA1GABRA5
SCHEMBL2628060 0.81 GABRA5 (0.44) GABRA1GABRA5
SCHEMBL286372 0.81 GABRA5 (0.44) GABRA1GABRA5
SCHEMBL286080 0.81 GABRA5 (0.44) GABRA1GABRA5
SCHEMBL286160 0.81 GABRA5 (0.42) GABRA1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed