SCHEMBL286463

SCHEMBL286463

CCCCc1noc(C)c1COc1cc(C(=O)OCC(N)=O)[nH]n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
LMNA P02545 2/20 0.34
GABRA1 P14867 3/20 0.33
GABRA5 P31644 2/20 0.33
L3MBTL1 Q9Y468 4/20 0.33
TDP1 Q9NUW8 1/20 0.33
KMT2A Q03164 3/20 0.33
GAA P10253 3/20 0.32
MEN1 O00255 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
TSHR P16473 2/20 0.32
CYP1A2 P05177 1/20 0.32
DPP4 P27487 1/20 0.32
ALPL P05186 2/20 0.32
HCRTR1 O43613 1/20 0.32
HTT P42858 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286460 0.88 ALPL (0.43) ALDH1A1GABRA5L3MBTL1KMT2AMEN1
SCHEMBL286582 0.87 KMT2A (0.38) ALDH1A1GABRA1GABRA5L3MBTL1KMT2A
SCHEMBL286328 0.87 KMT2A (0.38) ALDH1A1GABRA1GABRA5L3MBTL1KMT2A
SCHEMBL286337 0.86 HCAR2 (0.39) GABRA5L3MBTL1GAAALPLHTT
SCHEMBL286414 0.85 GABRA1 (0.32) ALDH1A1GABRA1GABRA5L3MBTL1KMT2A
SCHEMBL286160 0.82 GABRA5 (0.42) GABRA1GABRA5
SCHEMBL286161 0.82 POLB (0.40) GABRA1GABRA5L3MBTL1
SCHEMBL286143 0.81 ALDH1A1 (0.35) ALDH1A1LMNAGABRA1GABRA5L3MBTL1
SCHEMBL286394 0.81 L3MBTL1 (0.35) GABRA1GABRA5L3MBTL1
SCHEMBL286340 0.80 GABRA5 (0.44) GABRA1GABRA5ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163728-B2 Pyrazoles HOFFMANN-LA ROCHE INC. (US) 2012-04-24 US disclosed
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed