SCHEMBL28645581

SCHEMBL28645581

CC(C)c1cccc(Oc2ccccc2OC(C)(C)C(C)(C)O)c1.OBO

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.43
PTGS1 P23219 1/20 0.39
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36
CYP2D6 P10635 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC4 P56524 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
ALOX5 P09917 1/20 0.34
CETP P11597 2/20 0.34
BRAF P15056 1/20 0.34
PPARG P37231 3/20 0.33
LMNA P02545 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28633472 0.80 CETP (0.35) KDM4ETSHRMEN1KMT2ACETP
SCHEMBL28641325 0.80 L3MBTL1 (0.43) KDM4ECYP2D6KMT2AALDH1A1SMN1; SMN2
SCHEMBL29623492 0.78 CASP1 (0.43) CASP1PTGS1KDM4ETSHRMEN1
SCHEMBL28640739 0.77 MAPT (0.44) LMNAALDH1A1SMN1; SMN2L3MBTL1GAA
SCHEMBL25722842 0.74 HDAC4 (0.57) CASP1PTGS1KDM4ETSHRMEN1
SCHEMBL28925133 0.74 ALDH1A1 (0.42) CASP1KMT2ALMNAALDH1A1SMN1; SMN2
SCHEMBL28631825 0.74 LMNA (0.41) TSHRLMNAALDH1A1SMN1; SMN2
SCHEMBL28651923 0.72 RIPK1 (0.35) CASP1KDM4EMEN1KMT2APPARG
SCHEMBL13160048 0.71 AR (0.48) CASP1PTGS1KDM4ETSHRMEN1
SCHEMBL13255810 0.71 CASP1 (0.46) CASP1PTGS1KDM4ETSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493419-A EGFR tyrosine kinase inhibitor and application thereof 南京药石科技股份有限公司 2021-10-12 CN disclosed