SCHEMBL28758397

SCHEMBL28758397

CC(=O)OC(C)c1c(C)cc(C)cc1C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
ALDH1A1 P00352 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ACHE P22303 1/20 0.33
LMNA P02545 2/20 0.32
TAS1R3 Q7RTX0 2/20 0.32
TAS1R1 Q7RTX1 2/20 0.32
TAS1R2 Q8TE23 2/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962586 0.80 SLC6A2 (0.33) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL20102176 0.78 TSHR (0.35) TSHRHPGDNPSR1MCOLN3ALDH1A1
SCHEMBL27653319 0.78 TSHR (0.41) TSHRALDH1A1KDM4ECYP3A4CYP2C19
SCHEMBL13406762 0.74 L3MBTL1 (0.35) ALDH1A1KDM4ESLC6A2SLC6A4SLC6A3
SCHEMBL28599082 0.73 RAPGEF4 (0.36) ALDH1A1KDM4ECYP3A4CYP2C19SLC6A2
SCHEMBL16308869 0.72 LMNA (0.41) TSHRNPSR1ALDH1A1SLC6A2LMNA
SCHEMBL21342588 0.72 HTT (0.42) HPGDALDH1A1KDM4EACHELMNA
SCHEMBL334408 0.71 TSHR (0.34) TSHRHPGDALDH1A1KDM4ECYP3A4
SCHEMBL14490811 0.70 ALDH1A1 (0.38) HPGDNPSR1MCOLN3ALDH1A1KDM4E
SCHEMBL31607962 0.69 LMNA (0.47) TSHRALDH1A1CYP3A4ACHELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1780822-A Use of derivatives of 2, 4-dihydro- 1,2,4 triazole-3-thione as inhibitors of the enzyme myeloperoxidase (MPO) ASTRAZENECA AB (SE) 2006-05-31 CN disclosed