SCHEMBL2877908

SCHEMBL2877908

CCOC(=O)C1CCc2cccnc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.45
CYP2C19 P33261 2/20 0.44
MAPT P10636 5/20 0.44
KMT2A Q03164 4/20 0.44
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 3/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
MAPK1 P28482 3/20 0.41
RAB9A P51151 2/20 0.41
TP53 P04637 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALOX15 P16050 2/20 0.41
NPC1 O15118 1/20 0.41
CACNA1F O60840 1/20 0.41
NR1I2 O75469 1/20 0.41
GMNN O75496 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL883069 0.87 MAPT (0.56) HRH1CYP2C19MAPTKMT2AALDH1A1
SCHEMBL30557077 0.85 P2RX7 (0.39) HRH1MAPTKMT2AALDH1A1MEN1
SCHEMBL26120675 0.85 P2RX7 (0.39) HRH1MAPTKMT2AALDH1A1MEN1
SCHEMBL4166464 0.81 HTR2A (0.45) HRH1CYP2C19MAPTKMT2AALDH1A1
SCHEMBL2880939 0.80 OPRL1 (0.50) HRH1CYP2C19MAPTKMT2AALDH1A1
SCHEMBL2877889 0.80 MAPT (0.47) HRH1CYP2C19MAPTKMT2AALDH1A1
SCHEMBL27674615 0.79 KDM4E (0.40) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL2882382 0.79 HRH1 (0.43) HRH1CYP2C19MAPTKMT2AALDH1A1
SCHEMBL947365 0.79 ALDH1A1 (0.55) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL29683518 0.79 ALDH1A1 (0.55) MAPTKMT2AALDH1A1MEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4204401-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES Alterity Therapeutics Limited (AU) 2023-07-05 EP disclosed
CN-116323558-A Compounds and methods for treating diseases 艾特里提治疗有限公司 2023-06-23 CN disclosed
US-11603364-B2 Acyl hydrazone derivative compounds for treating disease Alterity Therapeutics Limited (AU) 2023-03-14 US disclosed
US-20220064142-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES ADJUVANT BIOTECHNOLOGY PTY LIMITED (AU) 2022-03-03 US disclosed
WO-2022040747-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES Alterity Therapeutics Limited (AU) 2022-03-03 WO disclosed
US-7855294-B2 Cycloalkanopyridine derivative BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-12-21 US disclosed
US-7855294-B2 Cycloalkanopyridine derivative BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-12-21 US disclosed
US-20070191419-A1 Cycloalkanopyridine derivative MSD K.K. (JP) 2007-08-16 US disclosed
US-20070191419-A1 Cycloalkanopyridine derivative MSD K.K. (JP) 2007-08-16 US disclosed
EP-1726590-A1 CYCLOALKANOPYRIDINE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-11-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11603364-B2 Acyl hydrazone derivative compounds for treating disease FH, ACOX1, HDAC1 HRH1 1107/4885CYP2C19 1836/4885MAPT 2903/4885
US-20220064142-A1 COMPOUNDS FOR AND METHODS OF TREATING DISEASES SLC30A6, SLC39A11, SLC40A1 HRH1 1792/4885CYP2C19 1708/4885MAPT 2397/4885
US-20070191419-A1 Cycloalkanopyridine derivative OPRL1, OPRK1, AVPR2 HRH1 2720/4885CYP2C19 3238/4885MAPT 287/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.