SCHEMBL28779148

SCHEMBL28779148

CC(C)(C)OC(=O)N1CCN(CC(=O)NCCCOCCOCCOCCCNC(=O)CCC(=O)O)CCN(C(=O)OC(C)(C)C)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
SIGMAR1 Q99720 4/20 0.40
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
ACKR3 P25106 3/20 0.39
TDP1 Q9NUW8 2/20 0.38
KEAP1 Q14145 2/20 0.37
NFE2L2 Q16236 2/20 0.37
STAT3 P40763 1/20 0.37
PKM P14618 1/20 0.36
ESRRB O95718 1/20 0.36
ESR1 P03372 1/20 0.36
ESRRA P11474 1/20 0.36
ESRRG P62508 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775091 0.90 ALDH1A1 (0.42) ALDH1A1KDM4ESIGMAR1TDP1
SCHEMBL28779145 0.86 CHRM2 (0.42) ALDH1A1SIGMAR1CHRM2CHRM4CHRM1
SCHEMBL15775094 0.85 KEAP1 (0.38) ALDH1A1KDM4EKEAP1NFE2L2PKM
SCHEMBL18533362 0.83 ACKR3 (0.43) SIGMAR1ACKR3KEAP1NFE2L2STAT3
SCHEMBL15047573 0.80 ALDH1A1 (0.45) ALDH1A1KDM4ESIGMAR1TDP1
SCHEMBL18471605 0.79 LMNA (0.43) SIGMAR1ACKR3KEAP1NFE2L2STAT3
SCHEMBL26419615 0.79 ALDH1A1 (0.46) ALDH1A1KDM4ESIGMAR1TDP1
SCHEMBL25510325 0.78 CACNA1H (0.46) ALDH1A1KDM4ESIGMAR1TDP1
SCHEMBL1509845 0.78 MEN1 (0.50) SIGMAR1TDP1
SCHEMBL15775309 0.77 ALB (0.37) ALDH1A1KDM4ESIGMAR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109320502-B Neurotensin receptor ligands 3B制药有限公司 2022-06-07 CN disclosed