SCHEMBL28790708

SCHEMBL28790708

Cc1ccccc1N1CCN(OC(=O)C(C)(C)C)CC1c1cccc(Br)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.36
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RIPK1 Q13546 2/20 0.33
CCR1 P32246 3/20 0.32
CCR2 P41597 2/20 0.32
HDAC1 Q13547 2/20 0.32
ROCK2 O75116 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SIGMAR1 Q99720 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
RECQL P46063 1/20 0.31
AR P10275 2/20 0.31
SCD5 Q86SK9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27828358 0.84 PKM (0.36) PDE5ATSHRNPSR1CCR1HDAC1
SCHEMBL1349076 0.82 HDAC6 (0.45) ROCK2LMNA
SCHEMBL27828433 0.80 PIK3C3 (0.37)
SCHEMBL28258134 0.74 TSHR (0.40) PDE5ATSHRNPSR1RIPK1ALDH1A1
SCHEMBL28046429 0.73 DRD2 (0.42) PDE5ATSHRNPSR1RIPK1ALDH1A1
SCHEMBL1349391 0.71 HDAC1 (0.46) PDE5AHDAC1MEN1KMT2ALMNA
SCHEMBL28018947 0.70 RIPK1 (0.49) NPSR1RIPK1ALDH1A1
Tert-Butyl Formate SCHEMBL28790709 0.69 HTR2C (0.38)
SCHEMBL28018952 0.68 RIPK1 (0.50) TSHRRIPK1ROCK2MEN1KMT2A
SCHEMBL1347787 0.67 NR1H2 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102056902-B Imidazolidine derivatives HOFFMANN LA ROCHE 2013-08-07 CN disclosed
CN-102056902-A Imidazolidine derivatives HOFFMANN LA ROCHE 2011-05-11 CN disclosed