SCHEMBL2880094

SCHEMBL2880094

CC(C)(C)NS(=O)(=O)c1ccc(-c2ccc(CC#N)cc2)s1.CC(C)(C)NS(=O)(=O)c1ccc(Br)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GALR3 O60755 1/20 0.39
RAB9A P51151 1/20 0.39
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PKM P14618 1/20 0.36
POLB P06746 1/20 0.35
THRB P10828 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
PRF1 P14222 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2087081 0.93 PKM (0.40) PKMPOLBPRF1MMP2MMP3
SCHEMBL620433 0.78 THRB (0.51) HTTLMNASMN1; SMN2GALR3RAB9A
SCHEMBL28291689 0.74 MMP2 (0.46) LMNASMN1; SMN2RAB9AALDH1A1MEN1
SCHEMBL7059253 0.73 PKM (0.39) HTTLMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL2089792 0.73 CA2 (0.52) PKM
SCHEMBL21124780 0.72 EDNRB (0.49) LMNASMN1; SMN2RAB9AALDH1A1MEN1
SCHEMBL2088655 0.67 PKM (0.38) HTTLMNARAB9AMEN1KMT2A
SCHEMBL1169197 0.66 SMN1; SMN2 (0.47) HTTLMNASMN1; SMN2GALR3RAB9A
SCHEMBL21084036 0.64 HPGD (0.44) LMNASMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL7736172 0.64 ALDH1A1 (0.39) LMNASMN1; SMN2RAB9AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227452-A2 PYRIDINE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2010-09-15 EP disclosed
WO-2009068468-A2 PYRIDINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2009-06-04 WO disclosed