SCHEMBL28801052

SCHEMBL28801052

CCOC(=O)CCNC(=O)C(Cc1ccccc1)C(=O)OC

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 2/20 0.58
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
NPY1R P25929 1/20 0.48
NPY2R P49146 1/20 0.48
POLB P06746 2/20 0.47
PKM P14618 1/20 0.46
LTA4H P09960 2/20 0.46
HRH4 Q9H3N8 1/20 0.45
PPID Q08752 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27874903 0.94 MMP8 (0.67) MMP8CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL7386752 0.84 CYP3A4 (0.51) MMP8CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL5496491 0.83 CYP3A4 (0.50) MMP8CYP3A4CYP2D6CYP2C19POLB
SCHEMBL5496496 0.83 CYP3A4 (0.50) MMP8CYP3A4CYP2D6CYP2C19POLB
SCHEMBL5495922 0.82 GPR142 (0.52) MMP8CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL5495924 0.82 GPR142 (0.52) MMP8CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL9560816 0.82 ALDH1A1 (0.50) MMP8CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL14503218 0.80 MMP8 (0.70) MMP8CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL7361284 0.80 LAP3 (0.64) MMP8CYP3A4CYP2D6CYP2C19POLB
SCHEMBL27546532 0.80 LAP3 (0.64) MMP8CYP3A4CYP2D6CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102712640-A Tricyclic heterocyclic compounds, compositions and methods of use thereof HOFFMANN LA ROCHE 2012-10-03 CN disclosed