SCHEMBL28824744

SCHEMBL28824744

Ic1ccc(C2CN2Cc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.44
MAPT P10636 1/20 0.41
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
SIGMAR1 Q99720 4/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
TP53 P04637 1/20 0.39
MDM2 Q00987 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
FUCA1 P04066 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824752 0.84 SIGMAR1 (0.50) OPRM1MAPTSIGMAR1
SCHEMBL28824734 0.83 RORC (0.52) OPRM1MAPTCYP3A4CYP2D6MAPK1
SCHEMBL28824755 0.79 LMNA (0.51) MAPTNR1H2NR1H3SIGMAR1CYP3A4
SCHEMBL28824750 0.79 OPRM1 (0.44) OPRM1MAPTNR1H2NR1H3SIGMAR1
SCHEMBL28824742 0.72 RORC (0.52) NR1H2NR1H3
SCHEMBL16226782 0.71 SIGMAR1 (0.55) NR1H2NR1H3SIGMAR1CYP1A2CYP3A4
SCHEMBL23870272 0.71 DPP4 (0.56) SIGMAR1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28824737 0.70 MAPT (0.45) MAPTSIGMAR1FUCA1
SCHEMBL24365249 0.70 MAPT (0.56) OPRM1MAPTNR1H2NR1H3SIGMAR1
SCHEMBL8659907 0.70 MEN1 (0.65) SIGMAR1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114941145-B Synthesis method of aziridine derivatives 天津理工大学 2023-08-18 CN disclosed
CN-114941145-A Synthetic method of aziridine derivative 天津理工大学 2022-08-26 CN disclosed