SCHEMBL28825568

SCHEMBL28825568

FC(F)(F)c1cccc([CH]c2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.46
FBP1 P09467 1/20 0.44
P4HB P07237 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GRIN1 Q05586 2/20 0.41
GRIN2B Q13224 2/20 0.41
TRPV4 Q9HBA0 1/20 0.41
DYRK1A Q13627 1/20 0.40
DYRK2 Q92630 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
TTR P02766 1/20 0.40
PIM1 P11309 1/20 0.40
CISD1 Q9NZ45 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237563 0.81 NFE2L2 (0.58) NFE2L2FBP1P4HBALDH1A1TTR
SCHEMBL28825622 0.78 NFE2L2 (0.56) NFE2L2FBP1P4HBALDH1A1L3MBTL1
SCHEMBL7435417 0.76 NFE2L2 (0.53) NFE2L2FBP1P4HBALDH1A1GRIN1
SCHEMBL28825569 0.76 NFE2L2 (0.46) NFE2L2FBP1P4HBL3MBTL1DYRK1A
SCHEMBL6205431 0.73 NFE2L2 (0.51) NFE2L2FBP1TTRPIM1CISD1
SCHEMBL16068085 0.72 GRIN1 (0.55) ALDH1A1L3MBTL1GRIN1GRIN2BMAOB
SCHEMBL543039 0.70 NFE2L2 (0.55) NFE2L2FBP1P4HBDYRK1ADYRK2
SCHEMBL13790316 0.70 NFE2L2 (0.82) NFE2L2FBP1P4HBCHRNB2CHRNB4
SCHEMBL18577798 0.69 NFE2L2 (0.50) NFE2L2FBP1P4HBPNMTMAOB
SCHEMBL23634792 0.69 KIF11 (0.63) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed