SCHEMBL28825637

SCHEMBL28825637

COc1cncc([CH]c2ccc(F)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.53
ROCK2 O75116 1/20 0.53
MAP4K4 O95819 1/20 0.53
PRKACA P17612 1/20 0.53
ROCK1 Q13464 1/20 0.53
DYRK1A Q13627 1/20 0.53
NTRK3 Q16288 1/20 0.53
PKN2 Q16513 1/20 0.53
CLK4 Q9HAZ1 1/20 0.53
MKNK2 Q9HBH9 1/20 0.53
STK17A Q9UEE5 1/20 0.53
NFE2L2 Q16236 7/20 0.49
CYP11B1 P15538 4/20 0.43
CYP11B2 P19099 4/20 0.43
EGFR P00533 1/20 0.40
PTGS1 P23219 1/20 0.40
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825596 0.84 ROCK2 (0.50) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL28696701 0.79 ROCK2 (0.46) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL28949613 0.78 CYP11B2 (0.51) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL14880245 0.78 NFE2L2 (0.76) NQO2NFE2L2RELA
SCHEMBL28825675 0.78 ROCK2 (0.50) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL28825560 0.77 CYP11B1 (0.44) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL14832276 0.76 S100B (0.45) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL14832275 0.76 S100B (0.45) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL28825677 0.76 GRIN1 (0.45) NQO2ROCK2MAP4K4PRKACAROCK1
SCHEMBL18240773 0.76 NFE2L2 (0.75) NQO2NFE2L2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed