SCHEMBL28825675

SCHEMBL28825675

COc1cncc([CH]c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.50
MAP4K4 O95819 1/20 0.50
PRKACA P17612 1/20 0.50
ROCK1 Q13464 1/20 0.50
DYRK1A Q13627 1/20 0.50
NTRK3 Q16288 1/20 0.50
PKN2 Q16513 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
STK17A Q9UEE5 1/20 0.50
CYP3A4 P08684 4/20 0.41
CYP2D6 P10635 2/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825617 0.84 GRIN2B (0.46) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825639 0.83 GRIN2B (0.44) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825596 0.78 ROCK2 (0.50) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825637 0.78 NQO2 (0.53) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL7975159 0.74 AHR (0.53) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL7974639 0.74 CHRM5 (0.46) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28696701 0.74 ROCK2 (0.46) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825677 0.74 GRIN1 (0.45) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL3298582 0.73 ALDH1A1 (0.64) CYP3A4ALDH1A1TP53MAPTAHR
SCHEMBL28949613 0.73 CYP11B2 (0.51) ROCK2MAP4K4PRKACAROCK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed