SCHEMBL28076582

SCHEMBL28076582

COc1ccc(CC(O)CN2CCC(Cc3ccc(OC)cc3N)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.55
DRD4 P21917 2/20 0.53
GAA P10253 1/20 0.49
GRIN2D O15399 1/20 0.49
GRIN3B O60391 1/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
GRIN1 Q05586 1/20 0.49
GRIN2A Q12879 1/20 0.49
GRIN2B Q13224 1/20 0.49
GRIN2C Q14957 1/20 0.49
GRIN3A Q8TCU5 1/20 0.49
HTR1A P08908 8/20 0.48
SLC6A4 P31645 8/20 0.48
ADRB2 P07550 1/20 0.47
ADRB1 P08588 1/20 0.47
ADRB3 P13945 1/20 0.47
MAPT P10636 1/20 0.45
ALOX12 P18054 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28076704 0.91 GAA (0.56) CYP2D6DRD4GAAGRIN2DGRIN3B
SCHEMBL28076624 0.86 HTR1A (0.52) DRD4GAAHTR1ASLC6A4ADRB2
SCHEMBL28076798 0.84 HTR1A (0.55) HTR1ASLC6A4RYR2
SCHEMBL28830809 0.82 DRD4 (0.62) CYP2D6DRD4GAAMAPT
SCHEMBL28830757 0.82 TSHR (0.60) CYP2D6DRD4GAA
SCHEMBL28076611 0.80 MAPT (0.48) DRD4GAAGRIN1GRIN2BHTR1A
SCHEMBL28076708 0.80 ADRA1A (0.49) DRD4GAAADRA1AHTR1ASLC6A4
SCHEMBL28076585 0.79 DRD4 (0.58) DRD4GAAADRB2ADRB1ADRB3
SCHEMBL28076620 0.78 HTR1A (0.46) DRD4GAAADRA1DADRA1AADRA1B
SCHEMBL3577962 0.76 RYR2 (0.49) HTR1ASLC6A4RYR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN claimed