SCHEMBL28831754

SCHEMBL28831754

COc1cc2c(cc1[N+](=O)[O-])OCC(=O)N2C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
PIK3CD O00329 2/20 0.38
PIK3R1 P27986 2/20 0.38
MTOR P42345 2/20 0.38
ALDH1A1 P00352 4/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 2/20 0.37
SIRT6 Q8N6T7 1/20 0.36
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
MAPT P10636 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
RAB9A P51151 2/20 0.34
CYP3A4 P08684 2/20 0.34
POLB P06746 1/20 0.34
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28831838 0.82 MAOB (0.36) TDP1PIK3CDPIK3R1MTORALDH1A1
SCHEMBL29847092 0.81 TDP1 (0.40) TDP1ALDH1A1LMNAHTTSIRT6
SCHEMBL4094748 0.79 TDP1 (0.42) TDP1ALDH1A1LMNAHTTSIRT6
SCHEMBL21468545 0.76 TDP1 (0.48) TDP1ALDH1A1LMNASIRT6KMT2A
SCHEMBL18937271 0.74 TERT (0.48) TDP1ALDH1A1LMNAHTTKMT2A
SCHEMBL16896891 0.74 L3MBTL1 (0.48) TDP1ALDH1A1HTTKMT2AMEN1
SCHEMBL28831852 0.72 SIRT6 (0.47) TDP1ALDH1A1LMNAHTTSIRT6
SCHEMBL3022688 0.70 ALDH1A1 (0.57) TDP1ALDH1A1LMNAHTTKMT2A
SCHEMBL16896874 0.69 MMP12 (0.44) TDP1ALDH1A1LMNAMAPTRAB9A
SCHEMBL15797122 0.68 MAPT (0.41) TDP1ALDH1A1LMNAHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115038707-B Azepine condensed ring compound and medical application thereof 中国医药研究开发中心有限公司 2024-11-22 CN disclosed
CN-115038707-A Azepine condensed ring compound and medical application thereof 中国医药研究开发中心有限公司 2022-09-09 CN disclosed