SCHEMBL28834853

SCHEMBL28834853

COC(=O)c1cc2c(ccn2-c2ccc(=O)n(C)c2)cc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.41
KDM4E B2RXH2 8/20 0.38
ALDH1A1 P00352 7/20 0.37
HSD17B10 Q99714 4/20 0.37
MAPT P10636 4/20 0.37
HPGD P15428 4/20 0.37
GAA P10253 3/20 0.37
GLA P06280 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
ATM Q13315 1/20 0.37
CFTR P13569 3/20 0.37
ABL1 P00519 1/20 0.36
TSHR P16473 2/20 0.36
ALOX15 P16050 1/20 0.36
NR4A2 P43354 3/20 0.35
BRD4 O60885 1/20 0.34
MYC P01106 1/20 0.34
NPC1 O15118 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28834826 0.83 SIRT6 (0.45) DGAT1KDM4EALDH1A1MAPTHPGD
SCHEMBL21231982 0.79 KDM4E (0.49) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL28834873 0.70 KDM4E (0.42) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL30184190 0.70 BRPF1 (0.49) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL23577596 0.70 BRPF1 (0.49) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL2924795 0.69 S100B (0.56) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL30326002 0.69 S100B (0.56) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL20595044 0.67 KDM1A (0.51) DGAT1KDM4EALDH1A1HPGDGAA
SCHEMBL25387340 0.67 BRPF1 (0.53) KDM4EALDH1A1HSD17B10BRD4RAB9A
SCHEMBL22140394 0.66 ALDH1A1 (0.53) KDM4EALDH1A1HSD17B10MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115028644-A SOS1 inhibitor heterocyclic compounds 首药控股(北京)股份有限公司 2022-09-09 CN disclosed