SCHEMBL28847907

SCHEMBL28847907

CC(=O)Oc1c(Cl)cc(C#N)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.39
AR P10275 2/20 0.39
GPR35 Q9HC97 3/20 0.38
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
LDHA P00338 1/20 0.35
LDHB P07195 1/20 0.35
AKR1B1 P15121 1/20 0.35
TTR P02766 1/20 0.35
ALB P02768 1/20 0.35
NCEH1 Q6PIU2 1/20 0.35
VCAM1 P19320 1/20 0.34
BACE1 P56817 1/20 0.34
MRGPRX4 Q96LA9 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28468360 0.79 TOP1 (0.47) GPR35LDHALDHBAKR1B1TTR
SCHEMBL4645395 0.78 ABCB11 (0.49) ABCB11BACE1POLBHTTMEN1
SCHEMBL23621178 0.78 MEN1 (0.48) ABCB11GPR35LDHALDHBAKR1B1
SCHEMBL5635782 0.77 ALDH1A1 (0.40) ABCB11LDHALDHBAKR1B1BACE1
SCHEMBL5688964 0.76 LMNA (0.43) ABCB11BACE1POLBHTTMEN1
SCHEMBL9575667 0.76 PDK1 (0.35) ARGPR35PDK1PDK2PDK3
SCHEMBL10551343 0.75 IMPDH2 (0.35) ABCB11ARGPR35LDHALDHB
SCHEMBL14659690 0.75 CYP19A1 (0.46) GPR35TTRALBBACE1POLB
SCHEMBL10787227 0.75 ABCB11 (0.42) ABCB11BACE1HTTALDH1A1
SCHEMBL4641540 0.75 POLB (0.43) ABCB11BACE1POLBHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107001278-A Tetrahydro isoquinoline derivative UCB生物制药私人有限公司 2017-08-01 CN disclosed