Thiophene

Thiophene

SCHEMBL28859237

C#CN(C(=O)OC(C)(C)C)c1ccccc1.c1ccsc1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.34
F2 P00734 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
AKT1 P31749 2/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSS P25774 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
BRD4 O60885 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GSK3B P49841 1/20 0.32
BCHE P06276 1/20 0.32
GBA1 P04062 1/20 0.32
HDAC3 O15379 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20759673 0.91 MEN1 (0.38) PAX8MEN1KMT2AAKT1RAB9A
SCHEMBL731186 0.73 ITGA4 (0.38) PAX8MEN1KMT2AL3MBTL1CYP3A4
SCHEMBL28905185 0.73 GBA1 (0.39) PAX8F2MEN1KMT2ARAB9A
SCHEMBL28506622 0.72 NPSR1 (0.39) PAX8MEN1KMT2ARAB9ANPSR1
SCHEMBL504005 0.70 L3MBTL1 (0.55) MEN1KMT2AAKT1RAB9ANPSR1
SCHEMBL8736767 0.70 MEN1 (0.43) PAX8MEN1KMT2AAKT1RAB9A
SCHEMBL3799516 0.70 L3MBTL1 (0.36) MEN1KMT2ARAB9ANPSR1L3MBTL1
SCHEMBL23113822 0.70 MEN1 (0.45) F2MEN1KMT2AL3MBTL1CYP3A4
SCHEMBL29903353 0.69 CHRM4 (0.36) MEN1KMT2ARAB9ANPSR1CTSL
SCHEMBL7200107 0.69 RAB9A (0.57) PAX8MEN1KMT2ARAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115043788-A Trifluoromethyl oxazole-2-ketone compound and preparation method and application thereof 南京工业大学 2022-09-13 CN claimed
CN-115043788-B Trifluoromethyl oxazol-2-one compound and preparation method and application thereof 南京工业大学 2023-10-20 CN disclosed
CN-115043788-A Trifluoromethyl oxazole-2-ketone compound and preparation method and application thereof 南京工业大学 2022-09-13 CN disclosed