SCHEMBL28880382

SCHEMBL28880382

Cc1c(Br)cccc1[C@@H](C)OC(N)=O

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.35
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
HCAR2 Q8TDS4 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
CXCL8 P10145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28880383 1.00 HTT (0.35) HTTCYP2C9CYP2C19CA12CA1
SCHEMBL11026259 0.85 HTT (0.44) HTTCYP2C9CYP2C19HCAR2ALDH1A1
SCHEMBL28880508 0.81 HTT (0.39) HTTCYP2C9CYP2C19MEN1KMT2A
SCHEMBL28880510 0.81 HTT (0.39) HTTCYP2C9CYP2C19MEN1KMT2A
SCHEMBL28880397 0.78 NPC1 (0.35) HTTCYP2C9CYP2C19MEN1KMT2A
SCHEMBL28880344 0.77 L3MBTL1 (0.35) LMNAALDH1A1
SCHEMBL28880345 0.77 L3MBTL1 (0.35) LMNAALDH1A1
SCHEMBL29163978 0.77 TAS2R14 (0.39) KMT2A
SCHEMBL29163979 0.77 TAS2R14 (0.39) KMT2A
SCHEMBL669484 0.76 ALDH1A1 (0.44) KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117940411-A Quinazoline derivative, or preparation method and application thereof 浙江海正药业股份有限公司 2024-04-26 CN disclosed
CN-117304182-A Compound with pyrimidohexa ring structure, pharmaceutical composition containing same and application of compound 上海海和药物研究开发股份有限公司 2023-12-29 CN disclosed
CN-116546985-A Pyridopyrimidine derivative and preparation method and application thereof 浙江海正药业股份有限公司 2023-08-04 CN disclosed
CN-115135315-A SOS1 inhibitors 米拉蒂治疗股份有限公司 2022-09-30 CN disclosed