SCHEMBL28880397

SCHEMBL28880397

Cc1c(Br)cccc1[C@@H](C)OC(=O)NC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CXCL8 P10145 1/20 0.34
HTT P42858 2/20 0.34
NLRP3 Q96P20 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 2/20 0.33
LPAR1 Q92633 1/20 0.33
ALPL P05186 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
SLC6A2 P23975 1/20 0.33
CHRNB4 P30926 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28880329 0.84 LPAR1 (0.37) NPC1RAB9AMEN1KMT2ACXCL8
SCHEMBL29163982 0.81 TAS2R14 (0.39) LMNALPAR1SMN1; SMN2
SCHEMBL30292599 0.80 SMN1; SMN2 (0.39) NPC1RAB9ACXCL8NLRP3ALDH1A1
SCHEMBL28880407 0.80 SMN1; SMN2 (0.39) NPC1RAB9ACXCL8NLRP3ALDH1A1
SCHEMBL28880362 0.78 SLC6A3 (0.35) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL28880383 0.78 HTT (0.35) MEN1KMT2ACXCL8HTTALDH1A1
SCHEMBL28880382 0.78 HTT (0.35) MEN1KMT2ACXCL8HTTALDH1A1
SCHEMBL25222548 0.76 KMT2A (0.47) NPC1RAB9AMEN1KMT2AHTT
SCHEMBL22497586 0.74 NPC1 (0.44) NPC1RAB9AMEN1KMT2AHTT
SCHEMBL17465167 0.74 HCAR2 (0.50) MEN1KMT2AHTTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999263-A SOS1 inhibitor with pyrido six-membered ring structure 上海海和药物研究开发股份有限公司 2024-05-07 CN disclosed
CN-115135315-A SOS1 inhibitors 米拉蒂治疗股份有限公司 2022-09-30 CN disclosed