SCHEMBL28880407

SCHEMBL28880407

Cc1c(C#N)cccc1[C@@H](C)OC(=O)NC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 1/20 0.36
SSTR4 P31391 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPK1 P28482 1/20 0.34
AAK1 Q2M2I8 1/20 0.34
NLRP3 Q96P20 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
MAOA P21397 1/20 0.33
HTR2B P41595 1/20 0.33
SOS1 Q07889 3/20 0.33
CXCL8 P10145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30292599 1.00 SMN1; SMN2 (0.39) SMN1; SMN2ALDH1A1KDM4ENPC1TP53
SCHEMBL29278098 0.86 SMN1; SMN2 (0.41) SMN1; SMN2ALDH1A1KDM4ENPC1TP53
SCHEMBL28880435 0.85 ALDH1A1 (0.38) SMN1; SMN2ALDH1A1KDM4ENPC1TP53
SCHEMBL28880397 0.80 NPC1 (0.35) SMN1; SMN2ALDH1A1NPC1RAB9ALMNA
SCHEMBL28880345 0.80 L3MBTL1 (0.35) SMN1; SMN2ALDH1A1LMNAL3MBTL1MAPK1
SCHEMBL28880344 0.80 L3MBTL1 (0.35) SMN1; SMN2ALDH1A1LMNAL3MBTL1MAPK1
SCHEMBL29163982 0.78 TAS2R14 (0.39) SMN1; SMN2LMNASOS1GAA
SCHEMBL23563447 0.74 TRPA1 (0.46) AAK1CTSLCTSBCTSK
SCHEMBL28880409 0.74 TRPA1 (0.46) AAK1CTSLCTSBCTSK
SCHEMBL29945842 0.74 TRPA1 (0.46) AAK1CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999263-A SOS1 inhibitor with pyrido six-membered ring structure 上海海和药物研究开发股份有限公司 2024-05-07 CN disclosed
CN-115135315-A SOS1 inhibitors 米拉蒂治疗股份有限公司 2022-09-30 CN disclosed