SCHEMBL28889233

SCHEMBL28889233

CCNC(=S)NC(=O)C(c1cccc(C)c1)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 2/20 0.41
ALDH1A1 P00352 6/20 0.39
KMT2A Q03164 5/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
ADRB2 P07550 1/20 0.39
MEN1 O00255 4/20 0.38
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PSEN1 P49768 3/20 0.37
PSEN2 P49810 3/20 0.37
APH1B Q8WW43 3/20 0.37
NCSTN Q92542 3/20 0.37
APH1A Q96BI3 3/20 0.37
PSENEN Q9NZ42 3/20 0.37
POLB P06746 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
NPSR1 Q6W5P4 3/20 0.36
ALOX12 P18054 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889342 0.90 OPRM1 (0.40) PHGDHALDH1A1KMT2ASMN1; SMN2ADRB2
SCHEMBL29941839 0.90 PHGDH (0.41) PHGDHALDH1A1KMT2AADRB2MEN1
SCHEMBL28889186 0.84 MEN1 (0.44) PHGDHALDH1A1KMT2ASMN1; SMN2ADRB2
SCHEMBL28889291 0.82 ADRB2 (0.39) PHGDHALDH1A1KMT2ASMN1; SMN2ADRB2
SCHEMBL29893566 0.82 ADRB2 (0.39) PHGDHALDH1A1KMT2ASMN1; SMN2ADRB2
SCHEMBL29942056 0.81 ALDH1A1 (0.43) ALDH1A1KMT2ASMN1; SMN2ADRB2MEN1
SCHEMBL28889200 0.80 ADRB2 (0.41) ALDH1A1KMT2ASMN1; SMN2ADRB2MEN1
SCHEMBL29941818 0.80 HDAC4 (0.41) PHGDHALDH1A1KMT2ASMN1; SMN2ADRB2
SCHEMBL28889196 0.79 TACR1 (0.43) ALDH1A1KMT2ASMN1; SMN2ADRB2MEN1
SCHEMBL28889226 0.79 AURKA (0.42) PHGDHALDH1A1KMT2AADRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed