SCHEMBL28889343

SCHEMBL28889343

COc1cccc(C(C(=O)NC(=S)NC2CC2)c2cc(C(F)(F)F)ccn2)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.42
HCRTR2 O43614 2/20 0.42
PHGDH O43175 1/20 0.38
SOS1 Q07889 1/20 0.37
MGLL Q99685 2/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
PDE4B Q07343 1/20 0.35
PDE4D Q08499 1/20 0.35
HTR1A P08908 2/20 0.35
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
DRD3 P35462 2/20 0.35
HTR2B P41595 2/20 0.35
GSK3B P49841 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889177 0.85 HDAC4 (0.40) PHGDHLMNAKMT2ANPSR1PDE4B
SCHEMBL28889234 0.84 PDE4B (0.38) PHGDHLMNAKMT2ANPSR1PDE4B
SCHEMBL29893652 0.84 PDE4B (0.38) PHGDHLMNAKMT2ANPSR1PDE4B
SCHEMBL29942052 0.83 KMT2A (0.40) HCRTR1HCRTR2PHGDHSOS1LMNA
SCHEMBL28889290 0.82 LMNA (0.40) PHGDHLMNAKMT2ANPSR1PDE4B
SCHEMBL28889330 0.82 ALDH1A1 (0.44) PHGDHLMNAKMT2ANPSR1ALDH1A1
SCHEMBL28889338 0.81 LMNA (0.41) HCRTR1PHGDHLMNAKMT2ANPSR1
SCHEMBL29893626 0.80 LMNA (0.41) HCRTR1PHGDHLMNAKMT2ANPSR1
SCHEMBL28889248 0.80 LMNA (0.41) HCRTR1PHGDHLMNAKMT2ANPSR1
SCHEMBL28889357 0.80 ALDH1A1 (0.39) PHGDHLMNAKMT2ANPSR1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed