SCHEMBL288942

SCHEMBL288942

CCCCOC(=O)N[CH]c1cccc2scnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.43
CYP1A2 P05177 4/20 0.43
CYP2C19 P33261 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
ALDH1A1 P00352 3/20 0.43
NPC1 O15118 3/20 0.43
NFKB1 P19838 1/20 0.43
STAT1 P42224 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 3/20 0.38
TGFBR1 P36897 1/20 0.37
CYP2C9 P11712 2/20 0.37
GAA P10253 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
PKM P14618 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288943 0.78 RAB9A (0.44) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL4704457 0.76 L3MBTL1 (0.44) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL3930322 0.69 TDP1 (0.58) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL7567608 0.69 CASP1 (0.44) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL7567614 0.68 RAB9A (0.34) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL3934013 0.66 NPC1 (0.53) RAB9ASMN1; SMN2ALDH1A1NPC1LMNA
SCHEMBL7221909 0.65 ALDH1A1 (0.41) ALDH1A1HSD17B10
SCHEMBL732122 0.65 ALDH1A1 (0.41) RAB9ASMN1; SMN2ALDH1A1NPC1L3MBTL1
SCHEMBL30565424 0.65 TSHR (0.53) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1
Benzo[D]Thiazole SCHEMBL28677081 0.64 LMNA (0.52) RAB9ACYP1A2CYP2C19SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427451-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BioLab Corporation (JP) 2012-03-14 EP disclosed
WO-2010128685-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BIOLAB CORPORATION (JP) 2010-11-11 WO disclosed