SCHEMBL28896263

SCHEMBL28896263

CCOC(=O)c1[nH]ccc1NC(CN)COC(F)C(F)F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.33
LMNA P02545 3/20 0.33
KMT2A Q03164 2/20 0.33
NUDT1 P36639 1/20 0.33
ALDH1A1 P00352 4/20 0.32
GAA P10253 3/20 0.32
POLB P06746 1/20 0.32
HTR6 P50406 1/20 0.32
CNR2 P34972 1/20 0.31
KDM4E B2RXH2 3/20 0.31
RAB9A P51151 2/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
RXFP1 Q9HBX9 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
MEN1 O00255 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29211269 0.83 KMT2A (0.34) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1
SCHEMBL28896499 0.82 SYK (0.38) KDM4EMAPTL3MBTL1
SCHEMBL28896261 0.82 KDM4E (0.34) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1
SCHEMBL28896837 0.80 SMN1; SMN2 (0.37) SMN1; SMN2LMNAKMT2AALDH1A1GAA
SCHEMBL28896253 0.77 NUDT1 (0.38) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1
SCHEMBL28896575 0.76 LMNA (0.33) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1
SCHEMBL24958271 0.73 SMN1; SMN2 (0.44) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1
SCHEMBL25241521 0.72 KDM4E (0.51) LMNAKMT2ANUDT1ALDH1A1GAA
SCHEMBL4200796 0.72 ALDH1A1 (0.45) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1
SCHEMBL1492325 0.70 KDM4E (0.50) SMN1; SMN2LMNAKMT2ANUDT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed