SCHEMBL28896273

SCHEMBL28896273

COc1ccc(CN(Cc2ccc(OC)cc2)CC(CBr)CC(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 2/20 0.48
TDP1 Q9NUW8 2/20 0.47
LDHA P00338 1/20 0.45
ACHE P22303 1/20 0.44
PTPN1 P18031 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
FFAR1 O14842 7/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
POLB P06746 1/20 0.43
TAS2R14 Q9NYV8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18942071 0.77 ALDH1A1 (0.54) TDP1LDHAACHEPTPN1ALDH1A1
SCHEMBL11221835 0.76 LDHA (0.66) LDHAFFAR1POLB
SCHEMBL28896648 0.75 TDP1 (0.44) NR1H3TDP1LDHAACHEPTPN1
SCHEMBL31392330 0.74 APLNR (0.45) ALDH1A1HTTSMN1; SMN2POLB
SCHEMBL11221992 0.73 LDHA (0.53) LDHAALDH1A1HTTSMN1; SMN2FFAR1
SCHEMBL27200631 0.73 MEP1B (0.60) LDHAACHEALDH1A1HTTSMN1; SMN2
SCHEMBL25401274 0.72 TDP1 (0.53) TDP1LDHAACHEALDH1A1HTT
SCHEMBL25401270 0.72 TDP1 (0.53) TDP1LDHAACHEALDH1A1HTT
SCHEMBL25241112 0.72 POLB (0.48) LDHAALDH1A1HTTSMN1; SMN2TSHR
SCHEMBL25225718 0.72 POLB (0.48) LDHAALDH1A1HTTSMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed