SCHEMBL28896648

SCHEMBL28896648

COc1ccc(CN(Cc2ccc(OC)cc2)CC(CBr)OC(C)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.44
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
HTT P42858 2/20 0.43
NR1H3 Q13133 2/20 0.43
TSPO P30536 1/20 0.43
LDHA P00338 1/20 0.42
APLNR P35414 1/20 0.41
ACHE P22303 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TSHR P16473 2/20 0.40
MAPK1 P28482 1/20 0.40
GSK3B P49841 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
MEP1A Q16819 1/20 0.39
MEP1B Q16820 1/20 0.39
PTPN1 P18031 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28959828 0.82 ALDH1A1 (0.39) TDP1ALDH1A1SMN1; SMN2HTTNR1H3
SCHEMBL28959827 0.80 TSPO (0.39) TDP1ALDH1A1SMN1; SMN2HTTNR1H3
SCHEMBL28896533 0.80 APLNR (0.38) TDP1ALDH1A1SMN1; SMN2HTTNR1H3
SCHEMBL28896273 0.75 NR1H3 (0.48) TDP1ALDH1A1SMN1; SMN2HTTNR1H3
SCHEMBL31392330 0.74 APLNR (0.45) ALDH1A1SMN1; SMN2HTTAPLNR
SCHEMBL25225718 0.72 POLB (0.48) ALDH1A1SMN1; SMN2HTTLDHAAPLNR
SCHEMBL25241112 0.72 POLB (0.48) ALDH1A1SMN1; SMN2HTTLDHAAPLNR
SCHEMBL4708637 0.72 LDHA (0.56) SMN1; SMN2HTTLDHATSHR
SCHEMBL14830786 0.71 NPC1 (0.41) ALDH1A1SMN1; SMN2HTTMEN1KMT2A
Acetic Acid SCHEMBL23429845 0.71 HRH3 (0.56) ALDH1A1SMN1; SMN2HTTTSPOLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-B 2-thio-2, 3-dihydropyrimidine-4-one derivatives, pharmaceutical compositions, preparation methods and applications thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed