SCHEMBL28896533

SCHEMBL28896533

COc1ccc(CN(Cc2ccc(OC)cc2)CC(CO[Si](C)(C)C(C)(C)C)OC(C)=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.38
TSHR P16473 4/20 0.37
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 1/20 0.36
NR1D1 P20393 1/20 0.36
TSPO P30536 1/20 0.36
KMT2A Q03164 2/20 0.36
NR1H3 Q13133 2/20 0.36
PTPN1 P18031 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
AR P10275 1/20 0.35
LDHA P00338 1/20 0.35
ACHE P22303 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28896201 0.81 POLB (0.47) APLNRTSHRALDH1A1KMT2AMEN1
SCHEMBL28896648 0.80 TDP1 (0.44) APLNRTSHRALDH1A1SMN1; SMN2HTT
SCHEMBL30029541 0.79 APLNR (0.40) APLNRALDH1A1SMN1; SMN2HTTNR1D1
SCHEMBL28959827 0.79 TSPO (0.39) TSHRALDH1A1SMN1; SMN2HTTTSPO
SCHEMBL28959828 0.78 ALDH1A1 (0.39) APLNRTSHRALDH1A1SMN1; SMN2HTT
SCHEMBL17391937 0.72 POLB (0.51) KMT2AARPOLB
SCHEMBL2177911 0.68 ADRB2 (0.46) ALDH1A1SMN1; SMN2HTT
SCHEMBL2177900 0.68 ADRB2 (0.46) ALDH1A1SMN1; SMN2HTT
SCHEMBL30406266 0.68 LTA4H (0.38) TSHRALDH1A1SMN1; SMN2KMT2ATDP1
SCHEMBL25439640 0.67 POLB (0.51) TSHRALDH1A1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-B 2-thio-2, 3-dihydropyrimidine-4-one derivatives, pharmaceutical compositions, preparation methods and applications thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed