SCHEMBL289080

SCHEMBL289080

O=C(Cl)Oc1cc2ccccc2o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 2/20 0.50
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 3/20 0.45
MAPT P10636 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CASP3 P42574 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
MAOB P27338 3/20 0.45
TSHR P16473 2/20 0.45
CA12 O43570 2/20 0.45
CA9 Q16790 2/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CA1 P00915 1/20 0.45
CA3 P07451 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4200612 0.84 FLT3 (0.52) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL27512860 0.83 FLT3 (0.47) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL3807363 0.82 KDM4E (0.51) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL10831738 0.82 FLT3 (0.55) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL8789115 0.82 FLT3 (0.50) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL11345699 0.81 HSD11B1 (0.51) KDM4EMAPTCA12CA9NPC1
SCHEMBL28346595 0.81 CA12 (0.49) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL31619040 0.81 MAPT (0.63) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL6607462 0.79 ALDH1A1 (0.53) FLT3KDM4EALDH1A1MAPTTDP1
SCHEMBL7461187 0.78 KDM4E (0.53) KDM4EALDH1A1MAPTTDP1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427451-B1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BIOLAB CO LTD (JP) 2019-03-20 EP disclosed
US-20180305373-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO Prism BioLab Co., Ltd. (JP) 2018-10-25 US disclosed
US-10017522-B2 Alpha helix mimetics and methods relating thereto Prism BioLab Co., Ltd. (JP) 2018-07-10 US disclosed
US-20150368262-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO Prism BioLab Co., Ltd. (JP) 2015-12-24 US disclosed
US-9040531-B2 Alpha helix mimetics and methods relating thereto Prism BioLab Co., Ltd. (JP) 2015-05-26 US disclosed
US-20120088770-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BIOLAB CORPORATION (JP) 2012-04-12 US disclosed
EP-2427451-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BioLab Corporation (JP) 2012-03-14 EP disclosed
WO-2010128685-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BIOLAB CORPORATION (JP) 2010-11-11 WO disclosed
CN-1203317-C Nano-colloidal gold marker immunization measurement method for testing carbofuran pesticide UNIV SHANGHAI JIAOTONG (CN) 2005-05-25 CN disclosed
CN-1445548-A Nano-colloidal gold marker immunization measurement method for testing carbofuran pesticide UNIV SHANGHAI JIAOTONG (CN) 2003-10-01 CN disclosed
EP-0160876-A1 1-Hetero-6-/1-Hydroxyethyl/-2-SR8-1-carbadethiapen-2-EM-3-carboxylic acids MERCK & CO. INC. (US) 1985-11-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150368262-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PLOD3, COL1A1, THPO FLT3 3898/4885KDM4E 4005/4885ALDH1A1 1511/4885
US-20120088770-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PLOD3, COL1A1, THPO FLT3 3898/4885KDM4E 4005/4885ALDH1A1 1511/4885
US-20180305373-A1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PLOD3, COL1A1, THPO FLT3 3898/4885KDM4E 4005/4885ALDH1A1 1511/4885
US-10017522-B2 Alpha helix mimetics and methods relating thereto PLOD3, COL1A1, THPO FLT3 3898/4885KDM4E 4005/4885ALDH1A1 1511/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.