SCHEMBL28908255

SCHEMBL28908255

COc1cc(Cl)ccc1OCc1cc(B(O)O)cs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.41
ENPP2 Q13822 1/20 0.41
KMT2A Q03164 3/20 0.40
NPC1 O15118 8/20 0.40
RAB9A P51151 7/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 1/20 0.38
ADRB2 P07550 1/20 0.38
POLB P06746 3/20 0.37
MAPT P10636 2/20 0.37
MITF O75030 1/20 0.37
UBE2N P61088 1/20 0.37
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PLK1 P53350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28520517 0.86 ACHE (0.44) ENPP2KMT2ANPC1RAB9AMEN1
SCHEMBL28521420 0.84 ALDH1A1 (0.45) MRGPRX4ENPP2KMT2ANPC1RAB9A
SCHEMBL28519536 0.81 USP2 (0.42) MRGPRX4ENPP2ALDH1A1MAPT
SCHEMBL28524257 0.79 ENPP2 (0.46) MRGPRX4ENPP2KMT2ANPC1RAB9A
SCHEMBL28530451 0.76 ENPP2 (0.43) ENPP2KMT2ANPC1RAB9AMEN1
SCHEMBL28519499 0.73 RXRA (0.40) ENPP2NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL29954639 0.72 ENPP2 (0.32) ENPP2POLB
SCHEMBL28521411 0.72 ENPP2 (0.51) MRGPRX4ENPP2ALDH1A1KDM4EPOLB
SCHEMBL28529096 0.70 NPC1 (0.42) ENPP2KMT2ANPC1RAB9AMEN1
SCHEMBL28520513 0.69 CA1 (0.41) ENPP2NPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602834-B Bruton's tyrosine kinase inhibitor 北京盛诺基医药科技股份有限公司 2021-01-08 CN disclosed