SCHEMBL28924400

SCHEMBL28924400

N#Cc1ccnc(-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.57
KMO O15229 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CTSK P43235 9/20 0.50
TGFBR1 P36897 1/20 0.47
KCNH2 Q12809 5/20 0.46
IDO1 P14902 1/20 0.46
GRIN1 Q05586 2/20 0.45
GRIN2B Q13224 2/20 0.45
GRM5 P41594 1/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CLK4 Q9HAZ1 1/20 0.44
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30081919 1.00 CTSS (0.57) CTSSKMOKDM4ECTSKTGFBR1
SCHEMBL893514 0.83 KIF11 (0.56) CTSSCTSKTGFBR1KCNH2
SCHEMBL9792939 0.82 CLK4 (0.62) IDO1GRM5CLK4
SCHEMBL17116600 0.81 CLK4 (0.51) IDO1GRM5CLK4
SCHEMBL6236184 0.79 CTSS (0.57) CTSSKMOKDM4ECTSKKCNH2
SCHEMBL3836507 0.79 CTSS (0.55) CTSSKDM4ECTSKGRIN1GRIN2B
SCHEMBL18535 0.78 CTSS (0.63) CTSSKMOCTSKKCNH2CTSL
SCHEMBL30158989 0.77 ASIC3 (0.53) TGFBR1GRM5CLK4
SCHEMBL2949191 0.77 ASIC3 (0.53) TGFBR1GRM5CLK4
SCHEMBL13692259 0.77 ABL1 (0.58) CTSSKMOKDM4ETGFBR1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403519-B Synthesis method of N-substituted isonicotinamide compound driven by visible light 河南师范大学 2024-03-01 CN disclosed
CN-115403519-A Synthesis method of N-substituted isonicotinamide compound driven by visible light 河南师范大学 2022-11-29 CN disclosed