Bicarbonate

Bicarbonate

SCHEMBL28930263

O=C([O-])[O-].OB(O)c1ccc(F)cc1.[K+].[K+]

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ORAI1 Q96D31 1/20 0.52
ORAI2 Q96SN7 1/20 0.52
ORAI3 Q9BRQ5 1/20 0.52
TRPV6 Q9H1D0 1/20 0.52
CA2 P00918 4/20 0.48
CA1 P00915 3/20 0.48
ENPP2 Q13822 3/20 0.43
KDM4E B2RXH2 1/20 0.41
MGLL Q99685 1/20 0.41
TSHR P16473 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
LPL P06858 1/20 0.41
LIPG Q9Y5X9 1/20 0.41
CXCR1 P25024 1/20 0.39
CXCR2 P25025 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508 0.85 ORAI1 (0.68) ORAI1ORAI2ORAI3TRPV6CA2
SCHEMBL21979751 0.85 ORAI1 (0.68) ORAI1ORAI2ORAI3TRPV6CA2
SCHEMBL18839425 0.83 ORAI1 (0.65) ORAI1ORAI2ORAI3TRPV6CA2
SCHEMBL31514900 0.80 LTA4H (0.55) ORAI1ORAI2ORAI3TRPV6CA2
SCHEMBL2551749 0.78 CA2 (0.61) ORAI1ORAI2ORAI3TRPV6CA2
Bicarbonate SCHEMBL28678657 0.77 ENPP2 (0.47) ENPP2KDM4EMGLLCES2CES1
Phenylboronic Acid SCHEMBL28664852 0.76 ENPP2 (0.70) ORAI1ORAI2ORAI3TRPV6CA2
Phenylboronic Acid SCHEMBL28610016 0.76 ENPP2 (0.70) ORAI1ORAI2ORAI3TRPV6CA2
SCHEMBL1668718 0.75 HSPB1 (0.56) ORAI1ORAI2ORAI3TRPV6CA2
SCHEMBL13806989 0.74 ORAI1 (0.54) ORAI1ORAI2ORAI3TRPV6CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108467370-B Triazole naphthoquinone bi-aromatic ring derivative or triazole naphthoquinone bi-aromatic heterocyclic derivative, and preparation method and application thereof 四川大学 2021-11-23 CN disclosed