SCHEMBL28940758

SCHEMBL28940758

CCc1cc(-c2cnns2)ccc1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.42
HSD17B1 P14061 3/20 0.39
IKBKB O14920 1/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37
GABRE P78334 1/20 0.37
GABRA6 Q16445 1/20 0.37
GABRG1 Q8N1C3 1/20 0.37
GABRG3 Q99928 1/20 0.37
GABRQ Q9UN88 1/20 0.37
MKNK1 Q9BUB5 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659243 0.81 ALDH1A1 (0.45) IKBKBMKNK1MKNK2ALDH1A1GAA
SCHEMBL28745316 0.74 PTPN1 (0.48) GPR52NEK2
SCHEMBL4996647 0.72 MKNK1 (0.50) MKNK1MKNK2ALDH1A1GAAMAPT
SCHEMBL2185846 0.72 HSD17B1 (0.42) GPR52HSD17B1GABRPGABRDGABRA1
SCHEMBL4437714 0.72 CHUK (0.59) HSD17B1IKBKBMKNK1MKNK2CDC7
SCHEMBL20113065 0.71 GPR52 (0.46) GPR52HSD17B1GABRPGABRDGABRA1
SCHEMBL16718767 0.70 ALDH1A1 (0.45) MKNK1MKNK2ALDH1A1GAAMAPT
SCHEMBL4109320 0.69 HSD17B1 (0.39) GPR52HSD17B1MKNK1MKNK2CDC7
SCHEMBL2659245 0.67 BCAT2 (0.49) IKBKBALDH1A1GAAMAPTHPGD
SCHEMBL11754806 0.67 HSD17B1 (0.51) HSD17B1ALDH1A1MAPTHTTGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1900080-A Inhibitors of cruzipain and other cysteine proteases AMURA THERAPEUTICS LTD (GB) 2007-01-24 CN disclosed
CN-1269822-C Inhibitors of kruenza protease and other cysteine proteases AMURA THERAPEUTICS LTD (GB) 2006-08-16 CN disclosed