SCHEMBL289465

SCHEMBL289465

COC(=O)c1ncc(Br)cc1CBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
OPRK1 P41145 13/20 0.39
NPSR1 Q6W5P4 1/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GMNN O75496 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
NFKB1 P19838 1/20 0.38
APEX1 P27695 1/20 0.38
GABRB3 P28472 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745103 1.00 CYP4F2 (0.40) CYP4F2CYP4A11OPRK1NPSR1TSHR
SCHEMBL30744962 0.89 OPRK1 (0.38) OPRK1NPSR1TSHRKDM4EGMNN
SCHEMBL20944537 0.89 OPRK1 (0.38) OPRK1NPSR1TSHRKDM4EGMNN
SCHEMBL22117014 0.85 TSHR (0.36) OPRK1NPSR1TSHRKDM4EGMNN
SCHEMBL24369751 0.83 OPRK1 (0.40) CYP4F2CYP4A11OPRK1NPSR1TSHR
SCHEMBL30402328 0.83 ALDH1A1 (0.40) CYP4F2CYP4A11NPSR1TSHRKDM4E
SCHEMBL29572125 0.83 MAPT (0.40) CYP4F2CYP4A11OPRK1NPSR1TSHR
SCHEMBL30849372 0.83 KDM4E (0.40) CYP4F2CYP4A11OPRK1NPSR1TSHR
SCHEMBL17544367 0.83 ALDH1A1 (0.40) CYP4F2CYP4A11NPSR1TSHRKDM4E
SCHEMBL18668409 0.83 MAPT (0.40) CYP4F2CYP4A11OPRK1NPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078119-A1 DEGRADER COMPOUNDS AND USES THEREOF BRISTOL MYERS SQUIBB CO (US) 2026-03-19 US disclosed
EP-4688771-A1 NOVEL FAK DEGRADER COMPOUNDS AND USES THEREOF Bristol-Myers Squibb Company (US) 2026-02-11 EP disclosed
US-12448368-B2 Indole compounds as androgen receptor modulators NIDO BIOSCIENCES, INC. (US) 2025-10-21 US disclosed
EP-3952870-B1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS NANJING ZENSHINE PHARMACEUTICALS CO LTD (CN) 2025-09-24 EP disclosed
US-12351570-B2 Disubstituted alkyne derivatives MERCK PATENT GMBH (DE) 2025-07-08 US disclosed
US-20250154107-A1 3,4-Dihydroisoquinolin-1(2H)-Ones Derivatives as STING Antagonists and the Use Thereof BEIGENE SWITZERLAND GMBH (CH) 2025-05-15 US disclosed
US-20250122176-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES INC (US) 2025-04-17 US disclosed
US-20250092021-A9 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES, INC. 2025-03-20 US disclosed
US-20250034134-A1 15-PGDH INHIBITOR AND USE THEREOF Wuhan Humanwell Innovative Drug Research and Development Center Limited Company (CN) 2025-01-30 US disclosed
US-20240408088-A1 PYRAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE ABBISKO THERAPEUTICS CO., LTD. (CN) 2024-12-12 US disclosed
US-20110053953-A1 AZA-Isoindolones and Their Use as Metabotropic Glutamate Receptor Potentiators - 613 ASTRAZENECA AB (SE) 2011-03-03 US disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed
US-20100286118-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 US disclosed
US-20100286118-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 US disclosed
US-20100286118-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 US disclosed
WO-2010129620-A1 IMIDAZO [ 1, 2 -A] PYRIDIN-2 -YL-PHENYL DERIVATIVES TO BE USED IN CANCER TREATMENT ALLA CHEM, LLC (US) 2010-11-11 WO disclosed
EP-2114940-A1 AZA-ISOINDOLONES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS - 613 AstraZeneca AB (SE) 2009-11-11 EP disclosed
WO-2008100715-A1 AZA-ISOINDOLONES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS - 613 ASTRAZENECA AB (SE) 2008-08-21 WO disclosed
WO-2008100715-A1 AZA-ISOINDOLONES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS - 613 ASTRAZENECA AB (SE) 2008-08-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286118-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 CNR1, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CNR2 CYP4F2 190/4885CYP4A11 138/4885OPRK1 270/4885
US-20240408088-A1 PYRAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE PRMT5, PRMT1, PRMT8 CYP4F2 177/4885CYP4A11 120/4885OPRK1 4725/4885
US-12351570-B2 Disubstituted alkyne derivatives BRCA1, MYC, PCNA CYP4F2 2833/4885CYP4A11 1749/4885OPRK1 4124/4885
US-20260078119-A1 DEGRADER COMPOUNDS AND USES THEREOF CTTN, SRC, PTK2 CYP4F2 4149/4885CYP4A11 3075/4885OPRK1 567/4885
US-20250122176-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS AR, FSHR, NR5A1 CYP4F2 3531/4885CYP4A11 1496/4885OPRK1 125/4885
US-20250034134-A1 15-PGDH INHIBITOR AND USE THEREOF HPGD, UGDH, PGD CYP4F2 135/4885CYP4A11 77/4885OPRK1 2213/4885
US-20110053953-A1 AZA-Isoindolones and Their Use as Metabotropic Glutamate Receptor Potentiators - 613 GRIN3A, GRM3, GRIN1 CYP4F2 1832/4885CYP4A11 914/4885OPRK1 332/4885
US-20250092021-A9 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS AR, FSHR, NR5A1 CYP4F2 3531/4885CYP4A11 1496/4885OPRK1 125/4885
US-12448368-B2 Indole compounds as androgen receptor modulators AR, FSHR, ADRB3 CYP4F2 3721/4885CYP4A11 1703/4885OPRK1 145/4885
US-20250154107-A1 3,4-Dihydroisoquinolin-1(2H)-Ones Derivatives as STING Antagonists and the Use Thereof STING1, IRF3, MAVS CYP4F2 4275/4885CYP4A11 3150/4885OPRK1 1842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.