SCHEMBL289682

SCHEMBL289682

CCOC(=O)c1nc(C)c(-c2cccs2)s1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.61
KDM4E B2RXH2 7/20 0.61
KMT2A Q03164 2/20 0.50
HPGD P15428 6/20 0.49
GAA P10253 5/20 0.49
CASP1 P29466 1/20 0.49
MAPT P10636 6/20 0.48
KEAP1 Q14145 1/20 0.48
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TSHR P16473 1/20 0.45
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
NPSR1 Q6W5P4 3/20 0.42
HIF1A Q16665 2/20 0.42
LMNA P02545 2/20 0.42
PPARG P37231 1/20 0.42
NCOA2 Q15596 1/20 0.42
NCOA1 Q15788 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6500653 0.79 ALDH1A1 (0.55) ALDH1A1KDM4EKMT2AHPGDGAA
SCHEMBL299236 0.78 MAPT (0.42) ALDH1A1KDM4EKMT2AHPGDMAPT
SCHEMBL5759200 0.78 ALDH1A1 (0.56) ALDH1A1KDM4EKMT2AHPGDGAA
SCHEMBL5761572 0.77 ALDH1A1 (0.55) ALDH1A1KDM4EKMT2AHPGDGAA
SCHEMBL290132 0.76 KDM4E (1.00) ALDH1A1KDM4EKMT2AHPGDGAA
SCHEMBL14380356 0.75 PTGS2 (0.51) KDM4EKMT2AGAAMAPTRAB9A
SCHEMBL3399928 0.75 CDC25B (0.49) ALDH1A1KDM4EKMT2AHPGDMAPT
SCHEMBL23079540 0.74 ALDH1A1 (0.52) ALDH1A1KDM4EKMT2AHPGDGAA
SCHEMBL290007 0.74 KDM4E (0.76) ALDH1A1KDM4EKMT2AHPGDGAA
SCHEMBL289663 0.74 JAK2 (0.47) ALDH1A1KDM4EKMT2AHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed