SCHEMBL28974658

SCHEMBL28974658

NS(=O)(=O)n1cccc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
APEX1 P27695 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28125877 0.80 POLB (0.41) POLBAPEX1TDP1L3MBTL1HDAC4
SCHEMBL17900455 0.77 PPME1 (0.49) POLBAPEX1TDP1L3MBTL1
SCHEMBL30599059 0.73 TSHR (0.44) POLBAPEX1TDP1L3MBTL1
SCHEMBL30599061 0.73 TSHR (0.44) POLBAPEX1TDP1L3MBTL1
SCHEMBL27851095 0.72 POLB (0.35) POLBAPEX1TDP1L3MBTL1HDAC4
SCHEMBL16540512 0.72 RAPGEF4 (0.56) POLBL3MBTL1
SCHEMBL8189051 0.71 ACLY (0.46) POLB
SCHEMBL782203 0.70
SCHEMBL8935030 0.69 ACLY (0.39) L3MBTL1
SCHEMBL14399002 0.69 FABP4 (0.36) POLBAPEX1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12544359-B2 1-aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors Infex Therapeutics Limited (GB) 2026-02-10 US disclosed
CN-119100967-A 1-Aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2024-12-10 CN disclosed
CN-119100967-A 1-Aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2024-12-10 CN disclosed
CN-119100967-A 1-Aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2024-12-10 CN disclosed
CN-114728902-B 1-Aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2024-09-13 CN disclosed
CN-114728902-B 1-Aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2024-09-13 CN disclosed
CN-116209652-A Synthesis of pyrrole acid derivatives 英菲克斯治疗有限公司 2023-06-02 CN disclosed
US-20230018460-A1 1-AMINOSULFONYL-2-CARBOXYPYRROLE DERIVATIVES AS METALLO-BETA-LACTAMASE INHIBITORS Infex Therapeutics Limited (GB) 2023-01-19 US disclosed
EP-4061800-A1 1-AMINOSULFONYL-2-CARBOXYPYRROLE DERIVATIVES AS METALLO-BETA-LACTAMASE INHIBITORS Infex Therapeutics Limited (GB) 2022-09-28 EP disclosed
EP-4061800-A1 1-AMINOSULFONYL-2-CARBOXYPYRROLE DERIVATIVES AS METALLO-BETA-LACTAMASE INHIBITORS Infex Therapeutics Limited (GB) 2022-09-28 EP disclosed
CN-114728902-A 1-aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2022-07-08 CN disclosed
CN-114728902-A 1-aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors 英菲克斯治疗有限公司 2022-07-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12544359-B2 1-aminosulfonyl-2-carboxypyrrole derivatives as metallo-beta-lactamase inhibitors CBR1, CBR3, SRR POLB 1356/4885APEX1 662/4885TDP1 4365/4885
US-20230018460-A1 1-AMINOSULFONYL-2-CARBOXYPYRROLE DERIVATIVES AS METALLO-BETA-LACTAMASE INHIBITORS CPN1, CMBL, ALDH7A1 POLB 1373/4885APEX1 408/4885TDP1 2584/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.