1-Methylxanthine

1-Methylxanthine

SCHEMBL29015259

CC(C)Cn1c(N)nc(=O)c2[nH]cnc21.Cn1c(=O)[nH]c2nc[nH]c2c1=O

nearest known ligand 0.57

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.57
ADORA2B P29275 9/20 0.57
PDE4A P27815 7/20 0.56
PDE4B Q07343 7/20 0.56
PDE4C Q08493 7/20 0.56
PDE4D Q08499 7/20 0.56
PDE2A O00408 3/20 0.56
PDE1A P54750 3/20 0.56
PDE1B Q01064 3/20 0.56
PDE1C Q14123 3/20 0.56
CFTR P13569 2/20 0.56
CYP1A2 P05177 2/20 0.56
PDE5A O76074 1/20 0.56
CYP3A4 P08684 1/20 0.56
TSHR P16473 1/20 0.56
MAPK1 P28482 1/20 0.56
ADORA1 P30542 1/20 0.56
SCN1A P35498 1/20 0.56
PDE6C P51160 1/20 0.56
PDE3B Q13370 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29015263 0.85 ADORA2A (0.61) ADORA2AADORA2BPDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL27663813 0.76 ADORA2B (0.77) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL60158 0.76 ADORA2A (0.70) ADORA2AADORA2BPDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL10996 0.76 ADORA2B (1.00) ADORA2AADORA2BPDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL9682658 0.74 ADORA2B (0.96) ADORA2AADORA2BPDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL28309011 0.74 ADORA2B (0.96) ADORA2AADORA2BPDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL27529726 0.74 ADORA2B (0.96) ADORA2AADORA2BPDE4APDE4BPDE4C
Isobutylmethylxanthine SCHEMBL7637581 0.73 PDE4A (0.94) ADORA2AADORA2BPDE4APDE4BPDE4C
Isobutylmethylxanthine SCHEMBL50315 0.72 PDE4A (1.00) ADORA2AADORA2BPDE4APDE4BPDE4C
Isobutylmethylxanthine SCHEMBL28814716 0.72 PDE4A (1.00) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096860-A Mammalian livestock pluripotent stem cell line from delayed embryo 阿塞尔塔有限公司 2023-05-09 CN disclosed