SCHEMBL2903225

SCHEMBL2903225

O=C(C=Cc1cccc(Cl)c1)N1CCC(=O)N(CCN2CCC(c3ccccc3)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
LMNA P02545 1/20 0.54
CCR2 P41597 11/20 0.52
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
KCNH2 Q12809 1/20 0.47
MAPT P10636 2/20 0.47
NPC1 O15118 1/20 0.47
HPGD P15428 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GPR183 P32249 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2903222 1.00 ALDH1A1 (0.54) ALDH1A1MEN1KMT2ALMNACCR2
SCHEMBL2903457 0.95 CCR2 (0.51) ALDH1A1MEN1KMT2ALMNACCR2
SCHEMBL2903456 0.95 CCR2 (0.51) ALDH1A1MEN1KMT2ALMNACCR2
SCHEMBL2905214 0.88 LMNA (0.73) ALDH1A1MEN1KMT2ALMNACCR2
SCHEMBL2905217 0.88 LMNA (0.73) ALDH1A1MEN1KMT2ALMNACCR2
SCHEMBL2904334 0.87 MEN1 (0.51) ALDH1A1MEN1KMT2ALMNADRD2
SCHEMBL2904336 0.87 MEN1 (0.51) ALDH1A1MEN1KMT2ALMNADRD2
SCHEMBL2903219 0.85 MAPT (0.51) ALDH1A1MEN1KMT2ALMNACCR2
SCHEMBL2903643 0.85 CCR2 (0.61) CCR2GPR183
SCHEMBL2903645 0.85 CCR2 (0.61) CCR2GPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed