SCHEMBL29033882

SCHEMBL29033882

COc1ccc(-c2cc(-c3ccc(C(=O)NC(C)c4ccc(N)cc4)cc3)n[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.54
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
MAPK1 P28482 3/20 0.54
CSNK2A2 P19784 1/20 0.49
CSNK2A1 P68400 1/20 0.49
LMNA P02545 4/20 0.49
ALDH1A1 P00352 2/20 0.49
TAS1R3 Q7RTX0 1/20 0.48
TAS1R1 Q7RTX1 1/20 0.48
CNR1 P21554 2/20 0.48
ROCK1 Q13464 6/20 0.46
ROCK2 O75116 5/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 3/20 0.46
PRKG1 Q13976 3/20 0.46
CYP2C9 P11712 2/20 0.46
PRKCG P05129 2/20 0.46
PRKACA P17612 2/20 0.46
RPS6KB1 P23443 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29033909 0.91 RAB9A (0.55) MAPTNPC1RAB9AMAPK1CSNK2A2
SCHEMBL29033888 0.89 PHGDH (0.45) MAPK1ROCK1ROCK2PRKG1CYP2C9
SCHEMBL29033874 0.88 BCHE (0.48) MAPTNPC1RAB9AMAPK1ALDH1A1
SCHEMBL29033886 0.83 PRKD1 (0.48) MAPK1ROCK1ROCK2PRKG1CYP2C9
SCHEMBL29033894 0.82 MAPT (0.53) MAPTNPC1RAB9AMAPK1ROCK1
SCHEMBL29033901 0.80 RAF1 (0.47) MAPTPHGDHKDM4ENPSR1PRKD1
SCHEMBL1608422 0.80 RAB9A (0.84) MAPTNPC1RAB9AMAPK1LMNA
SCHEMBL25309254 0.79 MAPT (0.53) MAPTNPC1RAB9AMAPK1CSNK2A2
SCHEMBL28354065 0.76 TAS1R3 (0.70) NPC1RAB9ALMNAALDH1A1TAS1R3
SCHEMBL16199794 0.75 RAB9A (0.75) MAPTNPC1RAB9AMAPK1CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394934-B Pyrazole benzamide compound as well as preparation method and application thereof 苏州大学 2023-06-13 CN disclosed
CN-114394934-A Pyrazole benzamide compound and preparation method and application thereof 苏州大学 2022-04-26 CN disclosed