SCHEMBL29065708

SCHEMBL29065708

COc1ccc(C23CC4CC(CC(C4)C2O)C3)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.47
P2RX7 Q99572 1/20 0.47
P2RX2 Q9UBL9 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
CNR2 P34972 2/20 0.46
MAOB P27338 2/20 0.44
MAOA P21397 1/20 0.44
HSD11B1 P28845 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 1/20 0.42
FAAH O00519 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607913 0.78 P2RX7 (0.40) EPHX2P2RX7CNR2HSD11B1LMNA
SCHEMBL12040557 0.75 LMNA (0.57) EPHX2P2RX7CNR2MAOBMAOA
SCHEMBL6901742 0.71 HSD11B1 (0.57) EPHX2P2RX7SIGMAR1CNR2MAOB
SCHEMBL8581921 0.70 CNR2 (0.63) EPHX2P2RX7P2RX2CNR2MEN1
SCHEMBL8064643 0.70 MEN1 (0.50) EPHX2P2RX2SIGMAR1CNR2SMN1; SMN2
SCHEMBL22027031 0.70 LMNA (0.40) P2RX7CNR2MAOBMAOAHSD11B1
SCHEMBL24241924 0.70 MEN1 (0.45) CNR2MAOBMAOAHSD11B1LMNA
SCHEMBL3844883 0.70 GAA (0.37) EPHX2P2RX7CNR2HSD11B1LMNA
SCHEMBL29287201 0.70 MEN1 (0.45) CNR2MAOBMAOAHSD11B1LMNA
SCHEMBL16352314 0.69 LMNA (0.56) MAOBMAOAHSD11B1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116789600-A Preparation method and application of novel tetrahydroindazole antitumor compound 深圳市人民医院 2023-09-22 CN claimed
CN-116444438-B Benzamide compound and preparation method, using method and application thereof 深圳市人民医院 2024-02-13 CN disclosed
CN-116789600-A Preparation method and application of novel tetrahydroindazole antitumor compound 深圳市人民医院 2023-09-22 CN disclosed
CN-116444438-A Benzamide compound and preparation method, using method and application thereof 深圳市人民医院 2023-07-18 CN disclosed