SCHEMBL29079309

SCHEMBL29079309

FC(F)(F)c1c[nH]c(-c2cccc(Br)n2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.45
GABRG2 P18507 2/20 0.45
GABRB3 P28472 2/20 0.45
GABRA3 P34903 2/20 0.45
HPGD P15428 1/20 0.33
NOTUM Q6P988 1/20 0.33
IDH1 O75874 6/20 0.33
IDH2 P48735 2/20 0.33
ALDH1A1 P00352 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
AHR P35869 1/20 0.31
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
PIM1 P11309 1/20 0.30
PIM3 Q86V86 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31138639 0.78
SCHEMBL9668609 0.77 HPGD (0.31) HPGD
SCHEMBL16534732 0.77 CBFB (0.47) GABRA1GABRG2GABRB3GABRA3HPGD
SCHEMBL25196015 0.74 SPR (0.39) GABRA1GABRG2GABRB3GABRA3ALDH1A1
SCHEMBL30442598 0.74 SPR (0.39) GABRA1GABRG2GABRB3GABRA3ALDH1A1
SCHEMBL22051478 0.74 CCR1 (0.39) GABRA1GABRG2GABRB3GABRA3
SCHEMBL10177266 0.73 DGAT1 (0.40) GABRA1GABRG2GABRB3GABRA3HPGD
SCHEMBL30442899 0.73 DGAT1 (0.40) GABRA1GABRG2GABRB3GABRA3HPGD
SCHEMBL31138525 0.73 ULK1 (0.32) KDM4E
SCHEMBL3795290 0.72 TRPA1 (0.35) HPGDNPSR1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116813619-A Macrocyclic inhibitors of Wee1 南京正大天晴制药有限公司 2023-09-29 CN disclosed