SCHEMBL29090285

SCHEMBL29090285

N#Cc1ccc(Sc2ncnc3c2CCNC3)c(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36
PNMT P11086 1/20 0.36
TRPV4 Q9HBA0 1/20 0.33
KDR P35968 2/20 0.32
AR P10275 4/20 0.32
HTR2C P28335 1/20 0.30
KCNH2 Q12809 1/20 0.30
CRHR1 P34998 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30603355 1.00 DRD2 (0.36) DRD2DRD3PNMTTRPV4KDR
SCHEMBL29329164 0.85 PTPN11 (0.38) KDRHTR2CKCNH2
SCHEMBL30603347 0.85 PTPN11 (0.38) KDRHTR2CKCNH2
SCHEMBL30603333 0.75 GPR119 (0.41)
SCHEMBL30603337 0.75 GPR119 (0.41)
SCHEMBL29330276 0.73 MAPK11 (0.36) PNMTHTR2CKCNH2
SCHEMBL29090312 0.72 TRPC5 (0.56) ARKCNH2
SCHEMBL29329546 0.70 MKNK1 (0.35) PNMT
SCHEMBL29330192 0.69 PTPN11 (0.38) HTR2C
SCHEMBL21002977 0.66 PNMT (0.34) DRD2DRD3PNMTHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116731013-A Heterocyclic compound, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2023-09-12 CN disclosed