SCHEMBL2922338

SCHEMBL2922338

COc1ccc(S(=O)(=O)N2[C@H](C(=O)NOC(=O)CCC3CCCC3)C[C@@H]3CCNC[C@@H]32)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 5/20 0.45
MMP2 P08253 3/20 0.45
MMP12 P39900 1/20 0.45
MMP1 P03956 7/20 0.43
MMP13 P45452 6/20 0.43
MMP3 P08254 4/20 0.42
MMP7 P09237 3/20 0.42
ALDH1A1 P00352 4/20 0.40
KLK7 P49862 2/20 0.40
EPHX2 P34913 1/20 0.39
ADAM17 P78536 1/20 0.39
KMT2A Q03164 1/20 0.38
TSHR P16473 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1656130 0.81 MMP1 (0.62) MMP9MMP2MMP12MMP1MMP13
SCHEMBL5532810 0.81 MMP1 (0.62) MMP9MMP2MMP12MMP1MMP13
SCHEMBL1656023 0.74 MMP9 (0.75) MMP9MMP2MMP12MMP1MMP13
SCHEMBL13201347 0.71 MMP9 (0.61) MMP9MMP2MMP12MMP1MMP13
SCHEMBL1656257 0.67 MMP9 (0.68) MMP9MMP2MMP12MMP1MMP13
SCHEMBL5532812 0.66 MMP1 (0.44) MMP9MMP1MMP13MMP3MMP7
SCHEMBL1655811 0.66 MMP9 (0.68) MMP9MMP2MMP12MMP1MMP13
SCHEMBL1655768 0.65 MMP2 (0.66) MMP9MMP2MMP12MMP1MMP13
SCHEMBL2927547 0.65 MMP9 (0.75) MMP9MMP2MMP12MMP1MMP13
SCHEMBL1656118 0.65 MMP9 (0.72) MMP9MMP2MMP12MMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768979-B1 OCTAHYDROPYRROLO[2, 3, C]PYRIDINE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCK SERONO SA (CH) 2010-09-29 EP claimed